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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T7477 | Antazoline | Others | |
Antazoline has antihistamine and anticholinergic effects.It used to treat a variety of arrhythmias. | |||
T16778 | Rocastine | AHR-11325 | Histamine Receptor |
Rocastine (AHR-11325) is a selective and potent non-sedating H1 receptor antagonist. | |||
T22713 | Decloxizine | Histamine Receptor | |
Decloxizine is a H1 receptor antagonist | |||
T7085 | Mebhydrolin | Mebhydroline | Histamine Receptor |
Mebhydrolin (Mebhydroline) is a specific histamine H1 receptor antagonist. | |||
T0263 | Chloropyramine hydrochloride | Nilfan,Alergosan,Halopyramine hydrochloride | FAK , VEGFR , Histamine Receptor |
Chloropyramine hydrochloride (Alergosan) is a histamine receptor H1 antagonist. | |||
T13352 | Wy 49051 | Wy-49051 | Histamine Receptor |
Wy 49051 is an orally active antagonist of H1 receptor(IC50 of 44 nM). | |||
T1469 | Levocetirizine | Levocetirizine HCl | Histamine Receptor |
Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a Histamine H1 Receptor Antagonist. | |||
T26253 | Tecastemizole | Norastemizole,R-43512,R43512,R 43512,T 1348 | Histamine Receptor |
Tecastemizole (R 43512) is a selective antagonist of H1 receptor and a major metabolite of astemizole with anti-inflammatory effects. | |||
T19966 | Clemastine | HS-592,Mecloprodin,Meclastin,HS592,HS 592 | Histamine Receptor |
Clemastine (Meclastin) is an antagonist of the H1 receptor and exhibits anti-inflammatory effects. | |||
T23297 | (S)-(+)-Dimethindene maleate | AChR , Histamine Receptor | |
(S)-(+)-Dimethindene maleate is an orally available, selective muscarinic M2 receptor and histamine H1 receptor antagonist that inhibits muscarinic M1, M3, and M4 receptors. | |||
T22354 | Levocetirizine Dihydrochloride | Xyzal Dihydrochloride,(-)-Cetirizine Dihydrochloride | Histamine Receptor |
Levocetirizine Dihydrochloride (Xyzal Dihydrochloride) is a third-generation peripheral H1-receptor antagonist. Acting as an antihistaminic agent, it specifically targets the histamine H1-receptor. Levocetirizine Dihydro... | |||
T17072 | Thiethylperazine dimaleate | Toresten,Thiethylperazine maleate,Norzine | Dopamine Receptor , Antibacterial , ABC , Histamine Receptor |
Thiethylperazine dimaleate (Thiethylperazine maleate) is an antagonist of the D2 receptor and H1 receptor. Thiethylperazine dimaleate is an activator of ABCC1 and possesses antimicrobial, anti-emetic, and antipsychotic e... | |||
T31488 | Dimethindene | Dimetindeno,Z 2001,Dimetindene,Z-2001,Z2001 | Potassium Channel , Endogenous Metabolite , AChR , Histamine Receptor |
Dimethindene (Dimetindeno) is a selective antagonist of H1 receptor and blocks K+ current. Dimethindene exhibits antihistamine and anticholinergic effects. | |||
T0445L | Promethazine hydrochloride | Promethazine HCl,Phenergan | Adrenergic Receptor , Histamine Receptor |
Promethazine hydrochloride (Promethazine HCl) , the first-generation antihistamine, is a strong antagonist of the H1 receptor and a moderate antagonist of the mACh receptor, moderate affinity for 5-HT2A, 5-HT2C, D2 and α... | |||
T83975 | Fenclozine Maleate | S 1429 | Histamine Receptor |
Fenclozine Maleate (S 1429) is a potential histamine H1 receptor antagonist , which can be used to study fever, inflammation and pain. | |||
T20884 | Hydroxyzine | Hydroxyzine free base | Histamine Receptor |
Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor. | |||
T1822 | Clemizole | HCV Protease , Histamine Receptor | |
Clemizole is an H1 histamine receptor antagonist, can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication. | |||
T1470L | Fexofenadine hydrochloride | Histamine Receptor | |
Fexofenadine Hydrochloride is a carboxylated metabolic derivative of terfenadine and long-lasting selective histamine H1 receptor antagonist, with antihistaminic activity. | |||
T10100 | QF0301B | 5-HT Receptor , Adrenergic Receptor | |
QF0301B is a potent α1-adrenergic receptor antagonist with inhibitory effects on α2-adrenergic receptors, 5-HT2A and histamine H1 receptors. | |||
T6405 | Bepotastine Besilate | Talion,TAU 284,Bepreve,Bepotastine Beslilate | Histamine Receptor |
Bepotastine Besilate (TAU 284) is a non-sedating and selective H1 receptor antagonist (pIC50: 5.7). |